Contrave

Bupropion · Naltrexone

Designed to target appetite regulation, this product is utilized to support weight control and alleviate behaviours associated with overeating.

Active ingredients
Bupropion · Naltrexone
Supply
Rx
Route
Oral use
Form
Prolonged-release tablet
Strengths
8/90mg

Contrave details

Condition
Obesity
Alternative names
Mysimba
Therapeutic class
Weight Loss Agent
Pharmacological class
Antiobesity Agent
Precautions and warnings
monitor blood pressure
Minor side effects
nausea; constipation; headache
Moderate side effects
dizziness; insomnia
Serious side effects
seizure, requires immediate medical attention
Dosage forms
Prolonged-release tablet
Administration route
Oral use
Supply category
Prescription only (specially controlled medicine)
Manufacturer
Orexigen Therapeutics
Onset Time
1–2 weeks
Duration
24 hours
Storage instructions
Store at room temperature.
Drug interactions
opioids; alcohol
Age restrictions
For adults only.
Pregnancy and breastfeeding
Pregnancy: Do not use. Breastfeeding: Do not use.
Contraindications

hypersensitivity to components; uncontrolled hypertension; seizure disorders; eating disorders

Patient summary

Designed to target appetite regulation, this product is utilized to support weight control and alleviate behaviours associated with overeating.

Mechanism of action

This combination medication acts by modulating the reward system and appetite-regulating centres in the brain to reduce food cravings and control caloric intake.

Where this medicine is registered

  • Singapore
  • Hong Kong
  • Thailand
  • Malaysia
  • Philippines
  • Indonesia
  • Taiwan
  • South Korea
  • Japan
  • Australia
  • New Zealand
  • UAE
  • South Africa

About Contrave

Contrave combines the active ingredients bupropion and naltrexone, a known pharmaceutical option for the management of obesity. Often sold under the brand name Mysimba, this medication is available as a tablet in a strength of 8/90mg. The manufacturer, Orexigen Therapeutics, developed this dual-action formulation to assist patients with weight control alongside a managed diet and physical activity programme.

Contrave availability in Asia

Contrave is registered across 11 markets including Thailand, Malaysia and the Philippines, with availability also in Taiwan, South Korea and the UAE. Generic variants of similar active ingredients, often manufactured in India, can offer a more budget friendly alternative to the original brand for expats living in regions with limited local stock. As with any treatment for obesity, this product is best used under a doctor’s care.