Methotrexate Tablets

Methotrexate

Utilized to manage autoimmune responses and indicated to alleviate inflammation-related tissue damage effectively.

Active ingredient
Methotrexate
Supply
Rx
Route
Oral use
Form
Tablet
Strengths
2.5mg

Methotrexate Tablets details

Alternative names
Maxtrex
Therapeutic class
Antimetabolite
Pharmacological class
Folic acid antagonist
Contraindications
severe hepatic impairment; pregnancy; breastfeeding; severe renal impairment
Precautions and warnings
regular blood monitoring required; photosensitivity precaution
Minor side effects
nausea; abdominal pain; fatigue
Moderate side effects
stomatitis; elevated liver enzymes
Dosage forms
Tablet
Administration route
Oral use
Supply category
Prescription only (specially controlled medicine)
Manufacturer
Hospira
Onset Time
3–6 weeks
Duration
long-term
Storage instructions
Store at room temperature in a safe place.
Drug interactions
alcohol; nsaids; salicylates
Age restrictions
Use with caution in elderly patients.
Pregnancy and breastfeeding
Pregnancy: absolute contraindication. Breastfeeding: contraindicated.
Serious side effects

bone marrow suppression, requires immediate medical attention; hepatotoxicity, requires immediate medical attention

Patient summary

Utilized to manage autoimmune responses and indicated to alleviate inflammation-related tissue damage effectively.

Mechanism of action

Methotrexate inhibits dihydrofolate reductase, thereby interfering with DNA synthesis and cellular replication to suppress overactive immune responses in chronic inflammatory conditions.

Where this medicine is registered

  • Singapore
  • Hong Kong
  • Thailand
  • Malaysia
  • Philippines
  • Indonesia
  • Taiwan
  • South Korea
  • Japan
  • Australia
  • New Zealand
  • UAE
  • South Africa

About Methotrexate Tablets

Methotrexate Tablets contain methotrexate, which is used for the management of Rheumatoid Arthritis, Psoriasis and Crohn’s Disease. This active ingredient is also marketed as Maxtrex. The medication is supplied as a tablet in the 2.5mg strength and is produced by manufacturers such as Hospira.

Methotrexate Tablets availability in Asia

Methotrexate Tablets are registered across 14 markets including the Philippines, Indonesia and Taiwan, with availability also in South Korea, Japan and the UAE. Generic versions of this medication, often sourced from India, provide a more affordable alternative to the original brand, supporting access for expats and patients living far from a standard medical supplier. This treatment is potent and should only be used under the direct supervision of a doctor.