Casodex

Bicalutamide

Designed to target tumour growth, indicated to manage advanced prostate cancer effectively.

Active ingredient
Bicalutamide
Supply
Rx
Route
Oral use
Form
Film-coated tablet
Strengths
50mg

Casodex details

Therapeutic class
Anti-Androgen
Pharmacological class
Non-steroidal Anti-Androgen
Contraindications
hypersensitivity to bicalutamide; pregnancy; women
Precautions and warnings
monitor liver function regularly; not indicated for use in children
Minor side effects
hot flushes; nausea; fatigue; constipation
Moderate side effects
gynaecomastia; breast tenderness; elevated liver enzymes
Dosage forms
Film-coated tablet
Administration route
Oral use
Supply category
Prescription only (specially controlled medicine)
Manufacturer
AstraZeneca
Onset Time
4–8 weeks
Duration
24 hours
Storage instructions
Store below 30°C.
Drug interactions
warfarin; ciclosporin
Age restrictions
Not for use in patients under 18.
Pregnancy and breastfeeding
Pregnancy: Not applicable (contraindicated). Breastfeeding: Not applicable.
Serious side effects

hepatitis, requires immediate medical attention; cholestasis, requires immediate medical attention

Patient summary

Designed to target tumour growth, indicated to manage advanced prostate cancer effectively.

Mechanism of action

Bicalutamide is a non-steroidal anti-androgen that binds to the androgen receptor. It prevents the binding of testosterone and dihydrotestosterone, thereby inhibiting the growth and progression of androgen-sensitive prostate cancer cells.

Where this medicine is registered

  • Singapore
  • Hong Kong
  • Thailand
  • Malaysia
  • Philippines
  • Indonesia
  • Taiwan
  • South Korea
  • Japan
  • Australia
  • New Zealand
  • UAE
  • South Africa

About Casodex

Casodex serves as a primary treatment for the management of advanced prostate cancer, utilizing bicalutamide as its active ingredient. This medication is produced by AstraZeneca and is supplied as 50mg tablets, offering a standard therapeutic choice for individuals managing this condition.

Casodex availability in Asia

Casodex is registered across 14 markets, including the UAE, Singapore and Hong Kong, with further availability in Thailand, Malaysia and the Philippines. Generic bicalutamide, notably manufactured in India, is often more affordable than the original brand for expats and people residing at a distance from a well-stocked medical outlet. This medication is best used under the direct care of a doctor.