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Afinitor

Everolimus

Developed to target cancer cells to support tumour growth suppression.

Active ingredient
Everolimus
Route
Oral use
Form
Tablet
Strengths
5 · 10mg

You will receive a quality generic equivalent, depending on stock.

Prescription rules on Afinitor vary by country.

Afinitor details

Therapeutic class
MTOR Inhibitor
Pharmacological class
Antineoplastic Agent
Contraindications
hypersensitivity to everolimus; hypersensitivity to sirolimus
Precautions and warnings
monitor blood glucose; risk of infection; regular blood count monitoring
Minor side effects
stomatitis; fatigue; rash
Moderate side effects
infections; pneumonitis; anaemia
Dosage forms
Tablet
Administration route
Oral use
Patient summary
developed to target cancer cells to support tumour growth suppression.
Supply category
Prescription only (specially controlled medicine)
Originator
Novartis
Onset Time
varies per patient
Duration
24 hours
Storage instructions
Store below 25°C. Protect from light.
Drug interactions
cytochrome p450 inhibitors; grapefruit
Pregnancy and breastfeeding
Pregnancy: must not be used. Breastfeeding: must not be used.
Serious side effects

interstitial lung disease, requires immediate medical attention; severe infections, requires immediate medical attention

Mechanism of action

Everolimus is a serine-threonine kinase inhibitor that acts as an mTOR inhibitor, reducing tumour cell proliferation and angiogenesis.

What you will receive

Afinitor is the originator brand name, made by Novartis. We use it here to identify the medicine only; we are not affiliated with Novartis and do not ship the original Afinitor.

  • You receive a generic equivalent: the same active ingredient (Everolimus) at the same dose, mostly recognised Indian branded generics from vetted manufacturers.
  • The exact brand supplied depends on what is in stock at the dispatching warehouse.
  • A regulated generic matches the original ingredient for ingredient by legal standard.

Are all generics really the same? Read the honest answer.

Where this medicine is registered

  • Singapore
  • Hong Kong
  • Thailand
  • Malaysia
  • Philippines
  • Indonesia
  • Taiwan
  • South Korea
  • Japan
  • Australia
  • New Zealand
  • UAE
  • South Africa

About Afinitor

Afinitor contains everolimus, a medication used to treat renal cell carcinoma, breast cancer and neuroendocrine tumours. This product is supplied as tablets in 5mg and 10mg strengths.

Afinitor availability in Asia

Afinitor is registered across 14 markets including Indonesia, Taiwan and South Korea, with availability also in Japan, the UAE and Singapore. Generic everolimus often provides an affordable alternative to the original brand for patients located far from a major pharmacy. This specialised medication is best used under a doctor’s care.