Hypercholesterolaemia

Hypercholesterolaemia means the level of LDL cholesterol in the blood is persistently high enough to raise the risk of coronary artery disease, heart attack, and stroke. It is one of the most common cardiovascular risk factors across East and Southeast Asia, where rapid dietary shifts towards processed and high-fat foods have driven rates sharply upward in countries including Singapore, Malaysia, Indonesia, and Thailand.

Medicines used to treat Hypercholesterolaemia

Lipitor

Atorvastatin

10 · 20 · 40mg

Indicated to manage high cholesterol levels and to alleviate the risk of future cardiovascular complications through HMG-CoA reductase inhibition.

From $0.43 / tablet View

Crestor

Rosuvastatin

5 · 10 · 20mg

Intended to target elevated cholesterol levels within the blood to manage cardiovascular risk.

From $1.24 / tablet View

Zocor

Simvastatin

5 · 10 · 20 · 40mg

Indicated to support the reduction of cholesterol levels, formulated to mitigate cardiovascular risk by inhibiting a key enzyme in cholesterol synthesis.

From $0.62 / tablet View

Livalo

Pitavastatin

1 · 2 · 4mg

Product indicated to manage hypercholesterolaemia and designed to support cardiovascular health by reducing cholesterol production.

From $0.76 / tablet View

Roszet

Rosuvastatin, Ezetimibe

10/10mg

Developed for hypercholesterolaemia, intended to target cholesterol synthesis and absorption to alleviate lipid levels and support cardiovascular health.

From $1.14 / tablet View

Questran

Colestyramine

4g

Indicated for hypercholesterolaemia, utilized to target bile acids in the gut to alleviate elevated blood cholesterol and support lipid management.

From $8.69 / sachet View

Zetia

Ezetimibe

10mg

Designed to support lipid management by reducing intestinal absorption of cholesterol.

From $1.13 / tablet View

Why cholesterol becomes a problem

Cholesterol itself is essential, but excess LDL particles deposit in artery walls, gradually narrowing them. Most people have no symptoms until a serious event occurs, so the condition is frequently discovered only during a routine blood test. A fasting lipid panel measures total cholesterol, LDL, HDL, and triglycerides and remains the standard way to confirm the diagnosis.

Genetics, diet, physical inactivity, obesity, and type 2 diabetes all contribute. Familial hypercholesterolaemia, an inherited form, produces very high LDL from early life and carries a substantially elevated lifetime risk if not treated.

Medicines used to lower LDL

Statins are the backbone of cholesterol management. They block an enzyme the liver uses to make cholesterol, reducing LDL by 30—55% depending on the agent and dose. Atorvastatin and rosuvastatin are high-potency statins used when larger reductions are needed, while simvastatin and pitavastatin suit moderate-risk profiles.

When statins alone are insufficient, ezetimibe can be added; it blocks cholesterol absorption in the gut rather than synthesis in the liver, and the two mechanisms together lower LDL more than either alone. Colestyramine is a bile acid sequestrant sometimes used in people who cannot tolerate statins.

Lifestyle alongside medicines

Diet changes and medicine work best together. Reducing saturated fat, increasing soluble fibre (oats, legumes, vegetables), and replacing refined carbohydrates with whole grains all contribute. Regular aerobic activity raises HDL and modestly lowers LDL. Smoking cessation improves overall cardiovascular risk beyond what medicine alone achieves. These changes do not eliminate the need for medicine in high-risk individuals, but they reduce the dose required and improve outcomes.